WebDec 1, 2024 · A series of N-(2-(3,4,5-trimethoxybenzyl)-benzoxazole-5-yl)benzamide derivatives (3a–3n) was synthesized and evaluated for its in vitro inhibitory activity against COX-1 and COX-2. The compounds with considerable in vitro activity (IC 50 < 1 µM), were evaluated in vivo for their anti-inflammatory and ulcerogenic potential. Out of the fourteen … WebEXAMPLE 3 34.8 g of 2,4-diamino-5- (3,4,5-trimethoxybenzyl)-pyrimidine and 97.2 g of triethyl orthoacetate are suspended in 240 ml of dimethylformamide and 1.2 ml of concentrated hydrochloric acid. The whole is stirred at 80 to 90 C. for 4 hours, treated with activated carbon and subjected to filtration, and the filtrate is concentrated in vacuo.
盐酸曲美他嗪 CAS:13171-25-0 广州硕谱生物科技有限公司
WebYou may be interested in these alternatives. Product Code. 11464384. 3,4,5-Trimethoxybenzyl alcohol, 98%, Thermo Scientific Chemicals. £78.60 / 50g. WebMar 31, 2011 · Two metal complexes of Co(II) and Cd(II) 5-(3,4,5-trimethoxybenzyl) pyrimidine-2,4-diamine (Trimethoprim) were synthesized and characterized by both analytical and spectroscopic methods. crow \u0026 moss chocolate
738-70-5 5-(3,4,5-Trimethoxybenzyl)pyrimidine-2,4-diamine Ambeed
WebAbstract. Radical-cation cyclodimerizations of electron-rich cyclic 1,3-dienes and radical-cation Diels-Alder reactions of these dienes with several electron-rich olefins have been investigated. In some cases the efficiency of the electron transfer could be increased if the electron acceptors were combined with LiClO 4 (special salt effect). WebApr 8, 2024 · Following a hybridization strategy, a series of 5-substituted-1H-indazoles were designed and evaluated in vitro as inhibitors of human monoamine oxidase (hMAO) A and B.Among structural modifications, the bioisostere-based introduction of 1,2,4-oxadiazole ring returned the most potent and selective human MAO B inhibitor (compound 20, IC 50 = … crow\u0027s auction gallery ltd